By H. Takagi, Hiroshi Takagi, Eric J. Simon
Advances in Endogenous and Exogenous Opioids includes the complaints of the foreign Narcotic learn convention (Satellite Symposium of the eighth overseas Congress of Pharmacology) held in Kyoto, Japan on July 26-30, 1981. The convention supplied a discussion board for discussing advances which were made within the figuring out of endogenous and exogenous opioids and tackled a wide range of issues starting from novel opiate binding websites selective for benzomorphan medications to the purification of opioid receptors and sequellae of receptor binding.
Comprised of 156 chapters, this booklet starts with an research of the interplay of opioid peptides and alkaloid opiates with mu-, delta-, and kappa-binding websites. The reader is then systematically brought to biochemical proof for kappa and sigma opiate receptors; the motion of morphine and oxymorphone as partial agonists at the field-stimulated rat vas deferens; mechanisms of supersensitivity within the enkephalinergic approach; and homes of the solubilized opiate receptor from human placenta. next chapters discover the biosynthesis of opioid peptides in addition to their localization, free up, and degradation; physiological and pharmacological activities of opioids; and using analgesia in acupuncture. result of behavioral and medical experiences of endogenous and exogenous opioids also are offered, and the structure-activity relationships of opioids are examined.
This monograph may be of curiosity to scholars, practitioners, and researchers within the fields of psychiatry and pharmacology.
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Extra resources for Advances in Endogenous and Exogenous Opioids. Proceedings of the International Narcotic Research Conference (Satellite Symposium of the 8th International Congress of Pharmacology) Held in Kyoto, Japan on July 26–30, 1981
RC and Zukin, RaS„ (1979) Proc0 Nat, Acad0 Sci. USA, 7£, 5372-5376. Kosterlitz, H C W. J. (1980) Proc. R. Soc 0 Lond 0 , 2^0, 113122. Zukin, R 0 S. RC (1981) Mol. G C , Thompson, J 0 A 0 , Huppler, R,E. and Gilbert, P 0 E 0 (1976) J. Pharmacol. Exp. , J^97, 517-532. (This work was supported by PHS grant DA-02575). S. R. J. A. SUMMARY A series of opioids have been used to study the opioid receptor in rat vas deferens. 3-Endorphin, etorphine, sufentanil and enkephalin behave as full ago nists in this preparation.
Chem. Pathol. and Pharmacol. 31, 173-176. 5. S. (1965) J. Med. Chem. 8, 609. 6. E. P. (1978) J. Med. Chem. 21, 598. , Tokyo SPECIFIC OPIATE BINDING SITES IN HUMAN PLACENTA A. Valette, G. Porthe", Y. Audigier", G. Pontonnier and J. Cros" INSERM, U. 168 Hopital La Grave, Toulouse and "CNRS Laboratoire de Pharmacologie et de Toxicologie Fondamentales 205. route de Narbonne, 31 078 TOULOUSE Cedex, France. SUMMARY Human placenta contains s p e c i f i c binding sites for 3 H-etorphine and 3,H-ethylketocyclazocine, which pharmacological characteristics correspond to the kappa receptors.
9218. J. and Aiello, E. (1976) Science, 104, 539. H. and Dvorkin, B. (1980) Science, in press. ). , Tokyo OPIOID RECEPTORS ON RAT MAST CELLS Y. Yamasaki, 0. Shimamura and H. Ijichi Second Department of Medicine, Kyoto Prefectural University of Medicine. Kamikyo-ku, Kyoto 602, Japan. SUMMARY Morphine was shown to reverse the inhibitory effect of PGE-, on IgE-mediated 14 C-serotonin release from rat mast cells dose-dependently, naloxone-antagonizably and stereospecifically. Met-enkephalin and p-endorphin mimicked such antiPGE-.
Advances in Endogenous and Exogenous Opioids. Proceedings of the International Narcotic Research Conference (Satellite Symposium of the 8th International Congress of Pharmacology) Held in Kyoto, Japan on July 26–30, 1981 by H. Takagi, Hiroshi Takagi, Eric J. Simon